PRL-8-53, le nootropic entsha, nayo eyaziwa ngegama layo imichiza imethyl 3- [2- [benzyl (imethyl) acid] ethyl] benzoate yi isongezelelo zokwenziwa nootropic. It yaphuhliswa-1970 nguGqirha uNikolaus Hansl e Creighton University Nebraska. Kuye kwafuneka ezinye izifundo yabantu elibonakalisa iimpendulo eyakhayo umsebenzi kwengqondo. Olunye uhlolisiso lubonisa ukuba i-compound sinokunceda ukubuyisa iinkumbulo elahlekileyo (hypermnesia).
Igama Product: PRL-8-53
Okunye Igama: imethyl 3- (2- (benzylmethylamino) ethyl) hydrochloride benzoate
3- (2-benzylmethylaminoethyl) benzoic acid methyl Ester hydrochloride
3- (2- (imethyl (phenylmethyl) acid) ethyl) benzoic acid methyl Ester hydrochloride
CAS Inombolo: 51352-87-5
Uvavanyo: 98%
Inkangeleko: powder White
Njani PRL-8-53 Work?
PRL-8-53 sisuka indibanisela benzoic acid kunye phenylmethylamine. Ubume imichiza wabumba yindibaniselwano ezi ziphumo khompawundi emibini ezimbaxa ukuba angasebenzisana receptors cholinergic, aqukiweyo modulating inkumbulo nokufunda iinkqubo ngaphakathi ebuchotsheni. PRL-8-53 yaziwa ukuba potentiate (ukwandisa impembelelo) dopamine kunye ngokungagqibelelanga zinqanda receptor serotonin. UGqr uNikolaus Hansl babekholelwa ukuba le nkangeleko isiphumo kungenza ukuba ukutshintsha kwemali eseleyo kwiinkqubo neurotransmitter CNS kwaye kukhokelela ekuphuculweni ukusebenza kwengqondo.
Kukho liye kuphela olunye uphando lwezonyango ebantwini eyenziweyo ukuvavanya ifuthe ichiza kwaye abonisa ukuphucuka kwinkumbulo ngomlomo, ixesha reaction ezibonwayo kunye nolawulo injini, ingakumbi abo phezu kweminyaka abantu 30. abadala badla ukuba bathobele ngakumbi memory kunye nokwehla kwengqondo, ngoko, inkumbulo kunye nezongezo ngcono cognitive zithande ukuba asebenze bhetele kuzo.
RPL-8-53 Imisebenzi:
Yandisa intelligence yengqondo
Ukukhulisa inkumbulo kunye namakhono ungqiyame
Ukuphucula amandla ingqondo ukusombulula iingxaki ukukhusela kuyo nayiphi imichiza okanye yokwenzakala emzimbeni
Ukunyusa izinga nezizathu
Ukwandisa ulawulo lwe mechanism zobuchopho subcortical / cortical
Ukuphucula siyazazi
Idosi imiphumela
Inkcazelo patent ekhoyo PRL 8-53 lubonisa iindidi 0.01-4mg / kg bodyweight. Noko ke, njengoko oko uluhlu elikhulu kunene, uluhlu oyinto 0.05-1.2 mg / kg. Oku kuthetha ukuba 3.4mg-81.6mg umntu 150 wesikiti kunye 4.55mg-109mg umntu 200 wesikiti. In kwetyala yabantu, akukho ziphumo bezingalindelekanga zirekhodwe; Noko ke, kunciphise umsebenzi motor kusaziwa iimpuku kunye neempuku xa unikwe ngeedosi enkulu PRL 8-53