J-147 foda

Takaitaccen Bayani:

J147 shine J-147 wani abu ne na musamman mai karfi, mai aiki da baki da kuma fili na neuroprotective yana da ikon haɓaka ƙwaƙwalwar ajiya a cikin dabbobin al'ada da kuma hana ƙarancin ƙwaƙwalwar ajiya a cikin cutar Alzheimer (AD) mice transgenic. Ayyukan neurotrophic da ƙwaƙwalwar ƙwaƙwalwar ƙwaƙwalwa na J-147 suna haɗuwa da karuwa a cikin matakan da aka samo neurotrophic factor (BDNF) da kuma bayyanar BDNF sunadaran amsawa, haɓaka LTP, adana furotin synaptic, raguwar amyloid plaques.

J-147 ne mai mahimmancin maganin neuroprotectant na baka wanda aka samo asali daga curcumin, kayan aiki mai aiki a cikin turmeric. Ba kamar curcumin ba, yana ketare shingen kwakwalwar jini cikin nasara sosai.

J-147 ne mai mahimmancin maganin neuroprotectant na baka wanda aka samo asali daga curcumin, kayan aiki mai aiki a cikin turmeric. Ba kamar curcumin ba, yana ketare shingen kwakwalwar jini cikin nasara sosai. Daga cikin su, J-147 yana aiki ta hanyar ɗaure zuwa ATP synthase. Yawan haɓakar ATP yana da alaƙa da tsarin tsufa. Bugu da ƙari, haɓaka matakan masu amfani da NGF da BDNF, J-147 na iya sarrafa wannan. Bugu da ƙari, J-147 yana hana monoamine oxidase B da kuma jigilar dopamine. Yana haɓaka haɓakar ƙwaƙwalwa ta hanyar haɓaka matakan haɓakar jijiyoyi (NGF) da abubuwan neurotrophic da aka samo daga ƙwaƙwalwa (BDNF). Mafi mahimmanci, J-147 na iya haɓaka haɓakar sabbin ƙwayoyin jijiya, haɓaka ƙwarewar koyo da ƙwaƙwalwar ƙwaƙwalwa, da haɓaka aikin fahimi.


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    Tags samfurin

    Sunan samfur:J-147 foda

    Wani Suna:2,2,2-Trifluoroacetic acid 1- (2,4-DiMethylphenyl)-2-[(3-Methoxyphenyl)Methylene]hydrazide],J-147,J147

    CAS No:1146963-51-0

    Matsakaicin: 99.0% Min

    Launi: Farin foda

    Shiryawa: 25kgs Ganguna

    Take:J-147 foda: Neuroprotective Agent for Alzheimer's Research & Anti-Aging Applications
    Bayanin Meta: Gano J-147 Foda, wani fili na neuroprotective curcumin wanda aka samu tare da ingantaccen inganci don haɓaka fahimi, ketare shingen kwakwalwar jini, da yin niyya ga cutar Alzheimer. Akwai a cikin ƙayyadaddun bayanai da yawa tare da jigilar kayayyaki na duniya.

    Babban Abubuwan Samfur

    1. Neuroprotective Powerhouse
      • Abun aiki na baka yana hana MAO-B (EC50 = 1.88 μM) da jigilar dopamine (EC50 = 0.649 μM)
      • Yana haɓaka ƙarancin spine dendritic da ƙwaƙwalwar ajiya a cikin berayen watanni 6 a 200ppm taro na abinci
      • Gwajin gwajin lokaci na asibiti na asibiti don Alzheimer ta Abrexa Pharmaceuticals & manyan cibiyoyi
    2. Multi-Target Anti-Tsofa Mechanism
      • Yana ɗaure zuwa ATP synthase don daidaita aikin mitochondrial
      • Yana ƙaruwa NGF/BDNF neurotransmitters yayin da yake toshe lalacewar ƙwayoyin kwakwalwa
      • Yana magance tsufa na jijiyoyin jini ta hanyar hana zubar jini na microvascular a cikin kwakwalwar linzamin kwamfuta
    3. Ƙididdiga na Fasaha
      • CAS No.: 1146963-51-0 | Tsarin kwayoyin halitta: C18H17F3N2O2
      • Tsafta: >99% | Solubility: 10 mM a cikin DMSO
      • Girman Girma: 1mg-500mg odar girma | 10mM/1mL bayani

    Jagora:

    1. Haɗin Kalma
      • Na farko: "Kariyar Neuroprotective", "Magungunan bincike na Alzheimer", "curcumin wanda aka samo asali"
      • Dogon wutsiya: "Mao-B mai hanawa don haɓaka fahimi", "tallafin mitochondrial anti-tsufa"
    2. Yarda da Fasaha na SEO
      • Ƙimar bayanan da aka tsara don abubuwan sinadarai (CAS, EC50, nauyin kwayoyin halitta)
      • Haɗin kai zuwa shafukan samfuri masu alaƙa (misali, abubuwan CAD-31, agonists na TrkB)
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    • Bayanin Tsaro: Ba a lura da cututtukan genotoxicity har zuwa 90μM a cikin gwaje-gwajen CeeTox

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