PRL-8-53, nootropic cusub, sidoo kale loo yaqaan by magaceeda kiimikada methyl 3- [2- [benzyl (methyl) amino] ethyl] benzoate waa dheeraadka ah synthetic nootropic. Waxaa la horumariyey ee 1970 ee Dr. Nikolaus Hansl at University Creighton ee Nebraska. Waxa uu lahaa qaar ka mid ah cilmiga aadanaha oo ay muujiyeen jawaabaha fiican in shaqada garashada. Mid ka mid ah daraasad muujisay in xarunta caawin kara dib u soo ceshano xusuus lumay (hypermnesia).
Product Name: PRL-8-53
Magaca Kale: methyl 3- (2- (benzylmethylamino) ethyl) hydrochloride benzoate
3- (2-benzylmethylaminoethyl) methyl acid Benzosyrene hydrochloride Ester
3- (2- (methyl (phenylmethyl) amino) ethyl) methyl acid Benzosyrene hydrochloride Ester
Number CAS: 51352-87-5
Isku dayo: 98%
Imaanshaha: budada White
Sidee ma PRL-8-53 Work?
PRL-8-53 waxaa laga darka of acid Benzosyrene iyo phenylmethylamine. Qaab dhismeedka kiimikada soo sameeyey isku dhafan oo ka mid ah laba natiijo oo xeryahooda ee xarunta a in la falgala receptors cholinergic, taas oo ay ku lug leeyihiin modulating xasuusta iyo barashada hababka maskaxda gudaheeda. PRL-8-53 waxaa sidoo kale loo yaqaan in ay potentiate (kordhiyo saamaynta) dopamine iyo qayb ahaan joogsada receptors serotonin. Dr. Nikolaus Hansl rumeysan yahay in profile saamayn this badan tahay keeni karto in ay wareeg ah dheelitirka ee nidaamka neurotransmitter habdhiska oo u wadin inuu soo hagaagay shaqaynta garashada.
Waxaa uu ahaa kaliya mid ka mid ah daraasad caafimaad oo aadanaha preformed si ay u qiimeeyaan saamaynta daroogada iyo waxa ay muujiyeen horumar ah ee xasuusta afka ah, waqtiga falcelinta muuqaal ah oo ay gacanta ku motor, gaar ahaan kuwa da'doodu ka weyn tahay 30. Dadka waaweyn waxa ay noqon ka badan ku xiran tahay xasuusta iyo hoos u dhac garashada, sidaas daraaddeed, xusuusta iyo supplements sii wanaajiyo garasho u muuqdaan in ay si fiican u shaqeeyaan iyaga on.
RPL-8-53 Functions:
In kor loo qaado sirdoonka maskaxda
Kor loogu xasuusta iyo awoodaha ku tiirsan
Hagaaji awooda maskaxda si ay u xaliyaan dhibaatooyinka iyo waxa ka kiimiko ah ama dhaawac jirka ah u ilaaliyaan
In kor loo qaado heerka dhiirogelin
In kor loo qaado ay gacanta of farsamo maskaxda cortical / subcortical
Hagaaji aragtida dareen
Qiyaasta iyo kooxda saamaynta
Macluumaadka patent diyaar u PRL 8-53 soo jeedinaya kala duwan oo 0.01-4mg / kg ee bodyweight. Si kastaba ha ahaatee, sida in uu yahay kala duwan oo aad u ballaaran, kala duwan oo ku haboon yahay 0.05-1.2 mg / kg. Arrintani waxay horseedaa in 3.4mg-81.6mg qof 150 pound ah oo 4.55mg-109mg qof 200 pound ah. In maxkamad aadanaha, waxyeelo ma laha waxa laga diiwaan geliyey, Si kastaba ha ahaatee, waxqabadka motor hoos lagu ogaadey jiirarka iyo jiirka marka siiyay xaddi badan oo PRL 8-53