Apigenin, as a known bioflavonoid, has been shown to exhibit various biological activities, including antioxidant, anti-inflammatory, antitumor, ant-genotoxic, anti-allergic, neuroprotective, cardioprotective, and antimicrobial.However, One of the most frequent sources of apigenin is celery (Apium graveolens), a marsh plant in the family of Apiaceae that has been cultivated as a vegetable since antiquity. Apigenin is the most extracted nutrient in celery, containing 108 mg apigenin per kg.Apigenin is one of the common dietary flavonoids, which is abundantly found in many fruits, vegetables, and medicinal herbs. It serves various physiological functions, such as antioxidant, potent anti-inflammatory, antiviral activities, antibacterial and blood pressure reduction.
Igoa oloa: aveese lau seleri Apigenin 98%
Latina Igoa: Apium graveolens L.
CAS leai: 520-36-5
Laau Vaega Faaaogaina: lau
Vaega: Apigenin
Assay: Apigenin 98,0% le HPLC
Valivali: Brown e samasama efuefu ma le uiga manogi ma tofo
GMO Tulaga: Free GMO
Teuina: i 25kgs drums fibre
Teuina: Tausi pusa tatalaina i mālū, nofoaga matutu, Ia o ese mai le malamalama malosi
Fata Olaga: O le 24 masina mai le aso o le tuuina
aafiaga Aneti-patu
taalo Apigenin se matafaioi taua i le puipuiga o le kanesa e ala i le faatauanau o apoptosis i laina eseese feaveai.
kanesa Ovarian:
na maua nisi suesuega e apigenin mafai ona taofiofia ai le tuputupu ae, proliferation, ma le fesiitaiga o CA-ov3 (feaveai kanesa ovarian tagata); e faatosina apoptosis o CA-ov3 e ala i le tausia o le stasis sela o le kanesa i G2 / vaega M. e fesootai ai le aafiaga i lea taimi ma inumaga.
kanesa Pancreatic:
Apigenin mafai ona taofiofia le proliferation o sela pancreatic kanesa. Apigenin starves le tuma i le faaitiitia o le puna o le suka, o le meaai i luga o lea kanesa sela ola. Gata i lea, e mafai ona faaleleia atili Apigenin le aoga o le togafitiga gemcitabine drug-.
Chemo-sensitization
Na iloa ai apigenin i mataupu maualalo sa a maualalo aafiaga cytotoxic ma le mafai ona faatosina leukemia myeloid matuitui tagata (hl-60) sela e apoptosis lelei. Ae peitai, apigenin mafai ona faaleleia ai le aafiaga inhibitory o cisplatin (DDP) i luga o hl-60 proliferation feaveai ao tuufaatasia ma concentrations eseese o DDP. Lea e mafai ona maua Apigenin aafiaga togafitiga-sensitization i hl-60; e mafai foi ona faaitiitia concentrations Low o apigenin le tetee o hl-60 sela i togafitiga-faaōleōle apoptosis, lea e mafai ona faatatau i le i lalo-tulafono faatonutonu o NF-κB ma BCL-2. (O NF-KB se ituaiga o porotini lavelave e pulea e tusitusiga DNA, o le tuuina atu o cytokines ma ola feaveai; ua encoded BCL2 i le tino e ala i le Gene BCL2, o le uluai tagata o le aiga BCL2 polotini faatonutonu e e mafai ona faatonutonu le oti feaveai)
puipuiga ate
e mafai ona faaitiitia ai le ate manua faaōleōle Apigenin e ischemia-reperfusion ala antagonizing lipid peroxidation ma scavenging radicals saoloto.
Apigenin mafai ona faaitiitia ate manuaga e mafua mai i le popole oxidative ona o lona antioxidant malosi ma gaoioiga aneti-inflammatory.
ua faamaonia o suesuega Pharmacological e apigenin ei ai se manino aafiaga e puipuia ai i le ava malosi-faaōleōle ate / manua hepatocyte, ma e fesootai lona auala autu i le inhibition o faaupuga CYP2E1 i le ate / hepatocyte.
taofia osteoporosis
Apigenin taofia osteoblastogenesis, osteoclastogenesis, ma e taofia ai foi leiloa ivi.
Apigenin puipuia o aano o ivi e faaitiitia leiloa ivi i le tino.
O nisi suesuega e faatatau i le MC3T3-E1, se laina feaveai vailaau osteoblast maua mai Mus musculus (isumu) calvaria, o loo maua e apigenin mafai ona taofiofia le TNF-α, IFN-γ, ona faaōleōle le secretion o ni cytokines e uunaia faavaeina osteoclast.
Apigenin inhibited foi le eseesega o 3T3-L1 sela vailaau adipose i adipocytes malosi, o lea inhibiting le eseesega auauna faaōleōle-eseesega inhibition adipocyte trovatore-6, MCP-1, oloa lectin.
Apigenin taofia le eseesega o osteoclasts mai RAW264.7 laina feaveai ma taofia i le faavaega o multinucleated osteoclasts. E mafai ona faatosina foi apoptosis osteoclast ma taofiofia resorption ivi.
Aneti-inflammatory ma aneti-oxidant gaoioiga
Apigenin restrains le faagasologa pupuga, e faateleina ai le trovatore-10 tulaga ma normalizes le faataamilosaga popole oxidative
Apigenin taofia cytokines fuafuaina e inflammatory ma faatosina tuuina cytokine le aneti-inflammatory.
O nisi o tusitusiga e taʻu mai ai apigenin alleviates pupuga pepa solo faaōleōle i le atuatuvale oxidative i le aano o le tino e modulating faailoga popole oxidative eseese, interleukins, maka enzyme le toto, ma le faailoaga o le tele o isi enzymes fesootai i ai.
Tulafono Faatonutonu o endocrine
Apigenin mafai ona faatonutonu toto suka, tausia thyroid le atoatoa ma pulea na maua peroxidation.It lipid e mafai ona faateleina ai le apigenin tulaga o inisalini ma thyroxine i manu suka, ma faaitiitia ai le faasalaga o le toto suka ma le gaoioiga o le kulukose-6-phosphorylase (G- 6-Pase).
Apigenin toe suia le aafiaga o le faateleina cholesterol serum, faateleina peroxidation lipid ate (LPO) ma faaitiitia gaoioiga o antioxidants e pei o catalase (pusi) ma superoxide dismutase (vaovao) i alloxan-faaōleōle manu.
I manu ma le suka masani toto, apigenin mafai foi ona faaitiitia serum cholesterol ma peroxidation lipid ate, ma faateleina ai le gaoioiga o antioxidants i sela.
meatotino Pharmacological o apigenin
ua faapipii Apigenin taua tele i le tausaga talu ai nei, o se faalauiloaina o le soifua maloloina aoga ona o lona maualalo toxicity vala aut ¯ u ma ona aafiaga o le soifua maloloina e aunoa versus sela o le kanesa, faatusatusa i le isi structurally fesootai flavonoids. Ua a tele o suesuega o faamatalaga molimau ua faaalia apigenin ua gafatia togafitiga tele mo le tele o faamai
galuega tauave:
-Inhibit le tuputupu ae o sela o le kanesa.
toto -Lower
-Protects le faiga cardiovascular
moe -Help, neura toafilemu, aveesea irritability
pupuga -Resist
osteoporosis -Prevent
aafiaga -Diuretic.
aggregation platelet -Inhibit.
talosaga:
-Medicine field, Health care field
nisi faamatalaga o TRB |
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R faamaoniga egulation | ||
USFDA, CEP, Kosher HALAL GMP Tusi faamaonia ISO | ||
Tulaga Aupito faatuatuaina | ||
Toeitiiti atoa le 20 tausaga, auina atu i fafo 40 atunuu ma itulagi, e sili atu nai lo le 2000 faaputuga gaosia e TRB e leai se faafitauli lelei, faagasologa o le faamamaina tulaga ese, e mama ma le mama pulea tatau USP, EP ma CP | ||
System Tulaga Auiliili | ||
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▲ System Inisiua Tulaga |
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▲ pulea Pepa o Faamatalaga |
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▲ System Aloaia |
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▲ Ofisa o Aoaoga |
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▲ Protocol Suetusi Lotoifale |
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▲ Ofisa o Suetusi Suppler |
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▲ System Fale Meafaigaluega |
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▲ Mea Ofisa o le Pulea |
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▲ o Oloa Gaosia Ofisa o le Pulea |
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▲ System Faaigoaina afifiina |
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▲ Falesuesue Ofisa o le Pulea |
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▲ faamaoniga System Aloaia |
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▲ Ofisa o Mataupu Tau le Va Faatonutonu |
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Pulea Punaoa Atoa ma Faagasologa | ||
Matua pulea mea mata uma, faaopoopoga ma afifiina materials.Preferred mata mea ma faaopoopoga ma pusa o loo afifi tuuina ma e tuuina mea mata US DMF number.Several pei faamautinoaga tuuina atu. | ||
Strong Faalapotopotoga Cooperative e lagolago | ||
Inisetiute o piolosi / Faalapotopotoga o microbiology / Academy o Saienisi ma Tekinolosi / Iunivesite |